平安! 发表于 2011-11-9 19:57
! s7 T& u4 C' a% O UPazopanib (100 mg/kg/day free base equivalent) 2 f1 H L- j9 e3 g. a" ?
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。
- u! Y E. T8 M! [6 p: C搜索了一下,原料一大堆。
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对不起!100mg/kg是用于移植瘤的,我弄错了。
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以下是正版说明书的推荐用量。/ F' n, A# b" W" \" U9 \/ C
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--------------------- DOSAGE AND ADMINISTRATION ----------------
" {. ~7 _+ j; g/ |+ ^( f; {0 _* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) # J7 R! B; H% m& z
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
Q c8 d0 V" |9 R& n---------------------DOSAGE FORMS AND STRENGTHS --------------
4 Q J* d) v0 k0 E- ^6 }200 mg tablets. (3)
' P$ K& Y+ A0 a6 e' s-------------------------------CONTRAINDICATIONS------------------------ |