平安! 发表于 2011-11-9 19:57 H. N! b V/ }; g4 Z/ U% Z+ P
Pazopanib (100 mg/kg/day free base equivalent) ( T% I( H2 `/ p0 J0 z. O, p* |; R
这是个已经在美国上市的老药了,能下载到正式药物使用说明书英文版。
7 h# M4 U! g* z搜索了一下,原料一大堆。
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9 `% l1 ?" G4 G: b! p. J6 P2 W对不起!100mg/kg是用于移植瘤的,我弄错了。) e/ m. w$ e) G! V' c/ z
, [5 g) P. i) d; E. y以下是正版说明书的推荐用量。
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. h( h j% b" c. k--------------------- DOSAGE AND ADMINISTRATION ----------------6 t- W8 b$ U1 L" u
* 800 mg orally once daily without food (at least 1 hour before or 2 hours after a meal). (2.1) # X* J+ W F. P, j- _0 \, c% B7 x
* Baseline moderate hepatic impairment – 200 mg orally once daily. Not recommended in patients with severe hepatic impairment. (2.2)
6 a! _# _4 l: H6 g---------------------DOSAGE FORMS AND STRENGTHS --------------
. A* G+ w8 _( b5 K- N( u: W200 mg tablets. (3)
& ?" }- ?8 n) Z- D# H. [-------------------------------CONTRAINDICATIONS------------------------ |